Microwave-assisted functionalization of bromo-fluorescein and bromorhodamine derivatives

Jin Wook Han, Juan C. Castro, Kevin Burgess

Research output: Contribution to journalArticle

41 Citations (Scopus)

Abstract

The overall goal of this project was to develop methodologies that would allow organometallic couplings of fluorescein and rhodamine derivatives. Consequently, borylation, Suzuki, and Sonogashira reactions of fragments derived from compounds 1 and 2 were investigated. Conventional and microwave heating were compared throughout the study.

Original languageEnglish
Pages (from-to)9359-9362
Number of pages4
JournalTetrahedron Letters
Volume44
Issue number52
DOIs
StatePublished - 2003 Dec 22

Fingerprint

Rhodamines
Microwave heating
Organometallics
Microwaves
Fluorescein
Heating
Derivatives

Keywords

  • Borylation
  • Fluorescent labels
  • Microwave acceleration of reactions
  • Sonogashira coupling
  • Suzuki coupling

Cite this

Han, Jin Wook ; Castro, Juan C. ; Burgess, Kevin. / Microwave-assisted functionalization of bromo-fluorescein and bromorhodamine derivatives. In: Tetrahedron Letters. 2003 ; Vol. 44, No. 52. pp. 9359-9362.
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Microwave-assisted functionalization of bromo-fluorescein and bromorhodamine derivatives. / Han, Jin Wook; Castro, Juan C.; Burgess, Kevin.

In: Tetrahedron Letters, Vol. 44, No. 52, 22.12.2003, p. 9359-9362.

Research output: Contribution to journalArticle

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